SCHEMBL6979174

SCHEMBL6979174

N#Cc1ccc(CCC(=O)N2CCCc3cc(C(=O)NCC4CCCCC4)ccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.50
NAMPT P43490 5/20 0.48
F10 P00742 2/20 0.45
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
DPP4 P27487 3/20 0.43
IDO1 P14902 1/20 0.42
KCNH2 Q12809 1/20 0.42
EGLN1 Q9GZT9 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6985092 0.87 F2 (0.51) F10OPRM1OPRD1OPRK1IDO1
SCHEMBL6984356 0.84 SMN1; SMN2 (0.53) TP53NAMPTHDAC1HDAC8HDAC6
SCHEMBL7409209 0.83 IDO1 (0.60) TP53HDAC1HDAC8HDAC6IDO1
SCHEMBL6977738 0.82 TP53 (0.51) TP53HDAC1HDAC8HDAC6IDO1
SCHEMBL6979412 0.82 NAMPT (0.49) TP53NAMPTHDAC1HDAC8HDAC6
SCHEMBL7085009 0.81 TP53 (0.49) TP53NAMPTHDAC1HDAC8HDAC6
SCHEMBL7948828 0.81 ITK (0.45) TP53HDAC1HDAC8HDAC6MEN1
SCHEMBL6981826 0.81 PDK1 (0.52) TP53HDAC1HDAC8HDAC6MEN1
SCHEMBL6985246 0.81 TP53 (0.51) TP53HDAC1HDAC8HDAC6IDO1
SCHEMBL7964635 0.80 TP53 (0.47) TP53HDAC1HDAC8HDAC6IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed