SCHEMBL7409209

SCHEMBL7409209

N#Cc1ccc(CCC(=O)N2CCCc3cc(C(=O)NCc4ccc(Cl)cc4)ccc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.60
KCNH2 Q12809 3/20 0.60
TP53 P04637 3/20 0.58
THRB P10828 2/20 0.47
HDAC1 Q13547 3/20 0.46
HDAC6 Q9UBN7 3/20 0.46
HDAC8 Q9BY41 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPT P10636 2/20 0.45
EGLN2 Q96KS0 1/20 0.44
USP30 Q70CQ3 1/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984356 0.85 SMN1; SMN2 (0.53) TP53HDAC1HDAC6HDAC8SMN1; SMN2
SCHEMBL6979174 0.83 TP53 (0.50) IDO1KCNH2TP53HDAC1HDAC6
SCHEMBL6981022 0.83 TP53 (0.51) IDO1KCNH2TP53THRBHDAC1
SCHEMBL6977738 0.83 TP53 (0.51) IDO1KCNH2TP53HDAC1HDAC6
SCHEMBL6984804 0.82 KCNH2 (0.45) IDO1KCNH2TP53HDAC1HDAC6
SCHEMBL6979412 0.82 NAMPT (0.49) TP53HDAC1HDAC6HDAC8SMN1; SMN2
SCHEMBL7958782 0.82 IDO1 (0.45) IDO1KCNH2TP53THRBHDAC1
SCHEMBL7085009 0.82 TP53 (0.49) IDO1KCNH2TP53HDAC1HDAC6
SCHEMBL6985246 0.81 TP53 (0.51) IDO1KCNH2TP53THRBHDAC1
SCHEMBL7958965 0.81 IDO1 (0.45) IDO1KCNH2TP53THRBHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed