SCHEMBL6979479

SCHEMBL6979479

CCC1(C(=O)O)CCC(N)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.33
ALDH1A1 P00352 1/20 0.32
GNAI3 P08754 1/20 0.32
GNAO1 P09471 1/20 0.32
GNAI1 P63096 1/20 0.32
OPRL1 P41146 1/20 0.32
FFAR3 O14843 1/20 0.31
SMYD3 Q9H7B4 1/20 0.31
GRM2 Q14416 2/20 0.31
GRM3 Q14832 2/20 0.31
GRM4 Q14833 2/20 0.31
CYP1A2 P05177 1/20 0.31
ALOX15 P16050 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GRM8 O00222 1/20 0.31
GRM6 O15303 1/20 0.31
LMNA P02545 1/20 0.31
GRM5 P41594 1/20 0.31
MTOR P42345 1/20 0.31
GRM1 Q13255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL385319 0.98 GNAI3 (0.34) CYP2C19ALDH1A1GNAI3GNAO1GNAI1
Hydrochloric Acid SCHEMBL385321 0.98 GNAI3 (0.34) CYP2C19ALDH1A1GNAI3GNAO1GNAI1
SCHEMBL1543252 0.88 ARG1 (0.35) CYP2C19ALDH1A1GRM2GRM3GRM4
SCHEMBL6802128 0.83 GNAI3 (0.32) GNAI3GNAO1GNAI1SMYD3
SCHEMBL17110192 0.83 GNAI3 (0.32) GNAI3GNAO1GNAI1SMYD3
SCHEMBL605108 0.81 CYP2C19 (0.34) CYP2C19ALDH1A1FFAR3LMNAMTOR
SCHEMBL1834809 0.81 CYP1A2 (0.36) CYP2C19ALDH1A1FFAR3CYP1A2ALOX15
SCHEMBL1066549 0.80 PLG (0.44) CYP2C19ALDH1A1LMNA
SCHEMBL245571 0.79
SCHEMBL30716833 0.79 CYP2C19 (0.42) CYP2C19ALDH1A1FFAR3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110494569-B Protease sensor molecules 联邦科学技术研究组织 2024-08-02 CN disclosed
US-11952612-B2 Protease sensor molecules COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2024-04-09 US disclosed
EP-3538665-B1 PROTEASE SENSOR MOLECULES PPB TECH PTY LTD (AU) 2024-01-03 EP disclosed
US-20190345535-A1 PROTEASE SENSOR MOLECULES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2019-11-14 US disclosed
EP-1244639-A4 2-CYCLOHEXYL BENZIMIDAZOLE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6495561-B2 TREATING MIGRAINE, DEPRESSION, ANXIETY, SCHIZOPHRENIA, PARKINSON'S DISEASE, OR STROKE MERCK & CO., INC. 2002-12-17 US disclosed
EP-1244639-A1 2-CYCLOHEXYL BENZIMIDAZOLE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-10-02 EP disclosed
US-20020055519-A1 2-cyclohexyl imidazopyridine NMDA/NR2B antagonists MERCK SHARP & DOHME CORP. 2002-05-09 US disclosed
US-6380205-B1 QUINAZOLINE THROUGH A C1-C4ALKYL, C1- C4ALKENYL, C1-C4ALKYNYL, C1-C4ALKOXY, AMINO, AMINOC1-C4ALKYL, HYDROXYC1-C4ALKYL, CARBONYL, CYCLOC3-C6ALKYL OR AMINOCARBONYL CHAIN, USEFUL FOR TREATMENT OF THE PAIN MERCK & CO., INC. 2002-04-30 US disclosed
US-20020032207-A1 2-Cyclohexyl quinazoline NMDA/NR2B antagonists MERCK & CO., INC. 2002-03-14 US disclosed
US-6291499-B1 TREATING MIGRAINE, DEPRESSION, ANXIETY, SCHIZOPHRENIA, PARKINSON'S DISEASE, OR STROKE MERCK & CO., INC. 2001-09-18 US disclosed
WO-2001032634-A1 2-CYCLOHEXYL BENZIMIDAZOLE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020055519-A1 2-cyclohexyl imidazopyridine NMDA/NR2B antagonists GRIN2C, GRIN1, GRIN3A CYP2C19 4060/4885ALDH1A1 2175/4885GNAI3 865/4885
US-20020032207-A1 2-Cyclohexyl quinazoline NMDA/NR2B antagonists GRIN2C, GRIN1, GRIN3A CYP2C19 3856/4885ALDH1A1 2927/4885GNAI3 570/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.