SCHEMBL6980044

SCHEMBL6980044

CCCC(CC(C)C)(C(=O)NN)C(=O)[C@](C)([C@H](C/C=C/c1ccccc1)C(=O)NO)N1C(=O)c2ccc(C)cc2C1=O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.36
GRIK1 P39086 1/20 0.30
GRIK2 Q13002 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982348 0.82 MMP1 (0.38) ADAM17GRIK1GRIK2
Hydrochloric Acid SCHEMBL6982151 0.78 CTSC (0.35) ADAM17GRIK1GRIK2
Hydrochloric Acid SCHEMBL6982639 0.76 CTSC (0.36) ADAM17GRIK1GRIK2
SCHEMBL6986163 0.75 ADAM17 (0.33) ADAM17
SCHEMBL6941953 0.74 ADAM17 (0.39) ADAM17GRIK1GRIK2
Hydrochloric Acid SCHEMBL6983018 0.72 CTSC (0.35) ADAM17GRIK1GRIK2
SCHEMBL6987148 0.72 CTSC (0.35) ADAM17GRIK1GRIK2
SCHEMBL6985245 0.72 ADAM17 (0.42) ADAM17
SCHEMBL6978290 0.72 EDNRB (0.30)
SCHEMBL6943076 0.71 ADAM17 (0.39) ADAM17GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed
EP-1089964-A1 HYDRAZINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2001-04-11 EP disclosed
WO-2000000465-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-01-06 WO disclosed