SCHEMBL6980246

SCHEMBL6980246

COC(=O)Oc1ccc2c(c1C)SCCC2(C)C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.36
RARB P10826 8/20 0.36
RARG P13631 7/20 0.36
PPARG P37231 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
JAK2 O60674 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RXRA P19793 3/20 0.31
CYP3A4 P08684 2/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971025 0.86 RARB (0.34) RARARARBRARGPTGS1PTGS2
SCHEMBL7998817 0.86 RARA (0.35) RARARARBRARGPPARGKDM4E
SCHEMBL7619004 0.78 RARA (0.42) RARARARBRARGPPARGPTGS1
SCHEMBL6970278 0.76 KDM4E (0.37) KDM4EHPGDHSD17B10JAK2ALDH1A1
SCHEMBL6971021 0.73 RXRA (0.39) RARARARBRARGPPARGPTGS1
SCHEMBL7831353 0.72 PTGDR (0.36) RARARARBRARGPTGS1PTGS2
SCHEMBL7501617 0.72 KDM4E (0.40) KDM4EHPGDHSD17B10JAK2ALDH1A1
SCHEMBL7809913 0.71 KDM4E (0.33) KDM4EHPGDHSD17B10JAK2ALDH1A1
SCHEMBL7624159 0.69 RARA (0.41) RARARARBRARGPPARGPTGS1
SCHEMBL7804185 0.69 KDM4E (0.36) KDM4EHPGDHSD17B10JAK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080089-B1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AG (DE) 2003-11-05 EP disclosed
EP-1080089-A1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2001-03-07 EP disclosed
WO-1999059991-A1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed