SCHEMBL6971025

SCHEMBL6971025

Cc1c(OC(=O)O)ccc2c1SCCC2(C)C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARB P10826 11/20 0.34
RARG P13631 11/20 0.34
RARA P10276 10/20 0.34
RXRA P19793 10/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
RXRB P28702 3/20 0.33
RXRG P48443 3/20 0.33
CYP26A1 O43174 3/20 0.33
CYP26B1 Q9NR63 2/20 0.33
CYP3A4 P08684 2/20 0.32
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980246 0.86 RARA (0.36) RARBRARGRARARXRAPTGS1
SCHEMBL7831353 0.85 PTGDR (0.36) RARBRARGRARARXRAPTGS1
SCHEMBL6971021 0.78 RXRA (0.39) RARBRARGRARARXRAPTGS1
SCHEMBL7619004 0.75 RARA (0.42) RARBRARGRARARXRAPTGS1
SCHEMBL6977102 0.75 MCL1 (0.31)
SCHEMBL7998817 0.72 RARA (0.35) RARBRARGRARARXRAPTGS1
SCHEMBL6981392 0.71 RXRA (0.33) RARBRARGRARARXRARXRB
SCHEMBL9197628 0.70 RARB (0.43) RARBRARGRARARXRARXRB
SCHEMBL7813372 0.70 KDM4E (0.38) KMT2A
SCHEMBL7496062 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080089-B1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AG (DE) 2003-11-05 EP disclosed
EP-1080089-A1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2001-03-07 EP disclosed
WO-1999059991-A1 PYRAZOLYLDIOXOTHIOCHROMANOYL DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed