SCHEMBL6980388

SCHEMBL6980388

Cc1cc(C(=O)OC(=O)c2ccoc2C)no1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 0.56
ALDH1A1 P00352 3/20 0.56
HPGD P15428 3/20 0.56
NPC1 O15118 11/20 0.42
RAB9A P51151 11/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
HTT P42858 3/20 0.42
TSHR P16473 1/20 0.42
POLB P06746 3/20 0.40
KMT2A Q03164 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
ESR1 P03372 1/20 0.40
ALOX12 P18054 1/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980382 0.79 PKM (0.58) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL8930043 0.73 ALDH1A1 (0.53) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL27759338 0.73 RAB9A (0.49) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL701960 0.70 HSD17B10 (0.59) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL1087642 0.70 MAPT (0.56) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL8267185 0.69 NPC1 (0.53) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL6972500 0.69 MAPT (0.50) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL18494022 0.69 RAB9A (0.50) PKMALDH1A1HPGDNPC1RAB9A
SCHEMBL434805 0.67 MEN1 (0.61) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL1757222 0.67 ALDH1A1 (0.60) PKMALDH1A1HPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218343-A4 PYRIDINE CARBOXAMIDE OR SULFONAMIDE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2003-06-18 EP disclosed
EP-1218343-A1 PYRIDINE CARBOXAMIDE OR SULFONAMIDE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-07-03 EP disclosed
WO-2001025203-A1 PYRIDINE CARBOXAMIDE OR SULFONAMIDE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-04-12 WO disclosed