SCHEMBL6980426

SCHEMBL6980426

N=C1CCCCC(C(CNC2=NCCC2)n2ccnc2)N1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.31
CYP17A1 P05093 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980113 0.73 CYP2D6 (0.33)
SCHEMBL6972299 0.71 TP53 (0.38)
SCHEMBL6964703 0.69 RAB9A (0.36) HSD17B10
Trifluoroacetic Acid SCHEMBL6979070 0.66 TP53 (0.36)
SCHEMBL6969171 0.64 CYP2D6 (0.40) ALOX15HSD17B10
SCHEMBL6969922 0.62 CYP2D6 (0.43) ALOX15HSD17B10
SCHEMBL6972842 0.61 CYP2D6 (0.46) ALOX15HSD17B10
SCHEMBL6978422 0.59 CYP19A1 (0.46) ALOX15
SCHEMBL19935934 0.55 CYP2D6 (0.59) ALOX15HSD17B10
SCHEMBL7622398 0.54 ALDH1A1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP claimed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US claimed
WO-1996033175-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1996-10-24 WO claimed
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed
WO-1996033175-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1996-10-24 WO disclosed