SCHEMBL6980522

SCHEMBL6980522

[N]C1CCCCC(Cc2cn(-c3ccccc3)nc2C(F)(F)F)N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 3/20 0.39
DGAT1 O75907 7/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
USP2 O75604 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ARF6 P62330 1/20 0.32
KCNH2 Q12809 2/20 0.31
DRD4 P21917 2/20 0.31
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
HTR2A P28223 1/20 0.31
HRH1 P35367 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974193 0.81 MPO (0.38) MPODGAT1KDM4EALDH1A1USP2
SCHEMBL6967526 0.81 MPO (0.38) MPODGAT1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL7088354 0.80 MPO (0.37) MPODGAT1KDM4EALDH1A1USP2
SCHEMBL6977100 0.73 KDM4E (0.31) KDM4EALDH1A1HRH1
SCHEMBL6978959 0.73 PTGS1 (0.42)
SCHEMBL6971234 0.70 MPO (0.35) MPODGAT1KDM4EALDH1A1MAPT
SCHEMBL6975255 0.70
SCHEMBL27722113 0.70 MPO (0.46) MPODGAT1KDM4EALDH1A1USP2
SCHEMBL6976719 0.68 POLB (0.59)
SCHEMBL6978425 0.68 CHRNB2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP claimed