SCHEMBL6977100

SCHEMBL6977100

[N]C1CCCCC(Cc2nc(C(F)(F)F)nn2-c2ccccc2)N1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31
TLR7 Q9NYK1 2/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HRH1 P35367 1/20 0.31
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967305 0.81 OPRL1 (0.36) ALDH1A1HTTLMNASMN1; SMN2CYP1A2
SCHEMBL6977098 0.81 CYP3A4 (0.31) TLR7NPC1LMNATP53PKM
SCHEMBL6978959 0.78 PTGS1 (0.42) NPC1LMNATP53PKMRAB9A
SCHEMBL6980522 0.73 MPO (0.39) KDM4EALDH1A1HRH1
SCHEMBL6974839 0.70 ALDH1A1 (0.41) KDM4EALDH1A1NPC1LMNATP53
SCHEMBL6980192 0.70 PTGS1 (0.31) SMN1; SMN2
SCHEMBL28869839 0.69 HRH1 (0.51) KDM4EALDH1A1GAAHTTTLR7
SCHEMBL6976719 0.68 POLB (0.59)
SCHEMBL6980592 0.67 FFAR1 (0.33)
SCHEMBL6976231 0.67 KDM4E (0.34) KDM4EALDH1A1GAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP claimed