SCHEMBL6980723

SCHEMBL6980723

Oc1cccc(CCCc2c[nH]nn2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.45
DRD1 P21728 2/20 0.45
TAAR1 Q96RJ0 1/20 0.45
CALM1 P0DP23 1/20 0.44
MGLL Q99685 1/20 0.42
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
OPRK1 P41145 2/20 0.41
ENPP2 Q13822 1/20 0.40
MIF P14174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31132412 0.83 HTR1B (0.45) DRD2DRD1TAAR1CHRM2CHRM1
SCHEMBL27892139 0.80 HTR2A (0.42)
SCHEMBL28221103 0.79 HTR2A (0.41)
SCHEMBL29869051 0.79 HTR2A (0.41)
SCHEMBL28368586 0.78 DRD2 (0.68) DRD2DRD1TAAR1CALM1MGLL
SCHEMBL31674607 0.78 DRD2 (0.68) DRD2DRD1TAAR1CALM1MGLL
SCHEMBL5048432 0.78 ESR1 (0.46) TAAR1CALM1MGLLCHRM2CHRM1
SCHEMBL2323457 0.76 DRD2 (0.65) DRD2DRD1TAAR1CALM1MGLL
SCHEMBL4949943 0.74 DRD2 (0.63) DRD2DRD1TAAR1CALM1MGLL
SCHEMBL966461 0.74 CALM1 (0.64) DRD2DRD1TAAR1CALM1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268473-A1 OXAZOLE DERIVATIVES AND THEIR USES AS TYROSINE KINASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 2003-01-02 EP disclosed
WO-2001077107-A1 OXAZOLE DERIVATIVES AND THEIR USES AS TYROSINE KINASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-10-18 WO disclosed