SCHEMBL6980736

SCHEMBL6980736

Cc1c(C)c2c(c(C)c1NC(=O)O)CC(C)(CN1CCC(CCNCCC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.38
MAOB P27338 2/20 0.38
TPSAB1 Q15661 2/20 0.34
KCNH2 Q12809 1/20 0.33
DPP4 P27487 1/20 0.33
CCR5 P51681 2/20 0.32
EPHX2 P34913 1/20 0.32
BCHE P06276 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983768 0.87 ACHE (0.35) ACHEMAOBTPSAB1KCNH2BCHE
Hydrochloric Acid SCHEMBL6976629 0.86 ACHE (0.35) ACHEMAOBTPSAB1BCHE
SCHEMBL6982741 0.82 ACHE (0.35) ACHEMAOB
Hydrochloric Acid SCHEMBL6984600 0.80 TPSAB1 (0.33) ACHEMAOBTPSAB1DPP4EPHX2
SCHEMBL6985682 0.77 SLC6A4 (0.49)
SCHEMBL6985715 0.75 KCNA3 (0.42)
SCHEMBL6985201 0.75 EPHX2 (0.45) TPSAB1EPHX2
Hydrochloric Acid SCHEMBL6978492 0.75 EPHX2 (0.45) EPHX2
SCHEMBL6986388 0.75 SLC6A4 (0.45) ACHEMAOBBCHE
Hydrochloric Acid SCHEMBL6982769 0.74 SLC6A4 (0.44) ACHEMAOBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed