SCHEMBL6980893

SCHEMBL6980893

CCOC(=O)Cc1ccccc1Nc1ccc2c(c1)CCCN2C(=O)CCc1ccc(C(=N)NC(=O)OC)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NOTUM Q6P988 1/20 0.37
ALDH1A1 P00352 4/20 0.37
LMNA P02545 3/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NR3C1 P04150 1/20 0.37
AVPR2 P30518 1/20 0.37
POLB P06746 2/20 0.36
KDM4E B2RXH2 1/20 0.35
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981558 0.92 NR3C1 (0.37) KMT2AMEN1MAPTSMN1; SMN2NOTUM
SCHEMBL6978185 0.79 ALDH1A1 (0.51) KMT2AMEN1MAPTSMN1; SMN2ALDH1A1
SCHEMBL6981262 0.78 NR3C1 (0.53) KMT2AMEN1MAPTSMN1; SMN2ALDH1A1
SCHEMBL6982230 0.78 NR3C1 (0.47) MAPTSMN1; SMN2ALDH1A1LMNAHPGD
SCHEMBL6979171 0.77 USP2 (0.41) MAPK1ALDH1A1LMNAHPGDNPSR1
SCHEMBL7960542 0.76 F2 (0.41) NPC1MAPTMAPK1RAB9ASMN1; SMN2
SCHEMBL6984100 0.76 TP53 (0.41) KMT2AMEN1NPC1MAPTMAPK1
Hydrochloric Acid SCHEMBL6985379 0.74 ALDH1A1 (0.42) NPC1MAPTMAPK1RAB9ASMN1; SMN2
SCHEMBL6987762 0.73 BRD4 (0.48) MAPTSMN1; SMN2ALDH1A1LMNAHPGD
SCHEMBL6985425 0.73 NR3C1 (0.52) KMT2AMEN1MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed