SCHEMBL6980928

SCHEMBL6980928

COC(=O)CN(C(=O)OC(C)(C)C)c1ccccc1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.38
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
STAT5B P51692 1/20 0.35
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA7 P43166 2/20 0.35
CA14 Q9ULX7 2/20 0.35
GSTO1 P78417 2/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
AKT1 P31749 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
F2 P00734 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257485 0.87 AKR1B1 (0.39) STAT5BCA1GSTO1CA2AKT1
SCHEMBL17077864 0.84 TSHR (0.39) LMNATSHRCA12CA1CA7
SCHEMBL7427088 0.83 MLYCD (0.39) MLYCDSTAT5BALDH1A1
SCHEMBL6906218 0.82 TSHR (0.40) MLYCDLMNATSHRCA12CA1
SCHEMBL6295798 0.81 MLYCD (0.48) MLYCDTSHRGSTO1AKT1ALDH1A1
SCHEMBL6907851 0.79 OPRM1 (0.43) MLYCDLMNATSHRCA12CA1
SCHEMBL31738254 0.79 KCNQ4 (0.33) LMNATSHRAKT1ALDH1A1HDAC3
SCHEMBL13258261 0.77 TDP1 (0.43) LMNATSHRCA12CA1CA7
SCHEMBL1826174 0.77 MLYCD (0.44) MLYCDCA12CA1CA7CA14
Hydrochloric Acid SCHEMBL6216388 0.75 MLYCD (0.43) MLYCDSTAT5BCA12CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289954-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
EP-1289950-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096296-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed
WO-2001096303-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed