SCHEMBL6980983

SCHEMBL6980983

Cc1[nH]c2ccccc2c1CC(=O)O.O=C(O)c1ccc(I)cc1

nearest known ligand 0.74

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.74
MAPT P10636 6/20 0.74
GAA P10253 4/20 0.74
ALDH1A1 P00352 3/20 0.74
CASP1 P29466 1/20 0.74
CASP7 P55210 1/20 0.74
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
EGFR P00533 2/20 0.50
AKR1C2 P52895 1/20 0.48
TSHR P16473 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 1/20 0.46
APEX1 P27695 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29612371 0.86 KDM4E (1.00) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL379103 0.86 KDM4E (1.00) KDM4EMAPTGAAALDH1A1CASP1
Hydrochloric Acid SCHEMBL1372439 0.85 KDM4E (0.97) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL4051892 0.79 PTPN5 (0.62) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL13401405 0.78 KDM4E (0.73) KDM4EMAPTGAAALDH1A1CASP1
Indole SCHEMBL28345849 0.75 KDM4E (0.76) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL5063952 0.74 ALDH1A1 (0.66) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL28092663 0.74 MAPT (0.76) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL15281758 0.74 MAPT (0.76) KDM4EMAPTGAAALDH1A1CASP1
SCHEMBL3384593 0.73 ATM (0.67) KDM4EMAPTGAAALDH1A1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218343-A4 PYRIDINE CARBOXAMIDE OR SULFONAMIDE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2003-06-18 EP disclosed
EP-1218343-A1 PYRIDINE CARBOXAMIDE OR SULFONAMIDE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-07-03 EP disclosed
WO-2001025203-A1 PYRIDINE CARBOXAMIDE OR SULFONAMIDE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-04-12 WO disclosed