SCHEMBL6981156

SCHEMBL6981156

O=C(CCCNC(=O)C1OC1C(=O)O)NC(=O)N1CCN(c2ccccc2Cl)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 9/20 0.44
DRD2 P14416 8/20 0.44
DRD4 P21917 6/20 0.42
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CACNA1G O43497 1/20 0.40
AKR1C3 P42330 1/20 0.40
HTR7 P34969 1/20 0.39
GFER P55789 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978349 0.84 GFER (0.55) DRD3DRD2DRD4ALDH1A1AKR1C3
SCHEMBL6978355 0.84 GFER (0.55) DRD3DRD2DRD4ALDH1A1AKR1C3
SCHEMBL6978386 0.79 KMT2A (0.49) DRD3DRD2DRD4ALDH1A1RAB9A
SCHEMBL6978390 0.79 KMT2A (0.49) DRD3DRD2DRD4ALDH1A1RAB9A
SCHEMBL6981803 0.73 ADAM10 (0.40) DRD3DRD2DRD4ALDH1A1AKR1C3
SCHEMBL6979020 0.72 SMN1; SMN2 (0.49) DRD3DRD2DRD4NPC1ALDH1A1
SCHEMBL6979028 0.72 SMN1; SMN2 (0.49) DRD3DRD2DRD4NPC1ALDH1A1
SCHEMBL27484010 0.71 GFER (0.50) ALDH1A1NPSR1HTR7GFERMAPT
SCHEMBL6981151 0.70 TGM2 (0.45) DRD3DRD2DRD4ALDH1A1AKR1C3
SCHEMBL6978563 0.70 CCR1 (0.50) ALDH1A1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6551999-B1 For therapy and prophylaxis of angiogenesis associated with wound healing, inflammation, growth of tumor and the like; angiogenesis as seen in diabetic retinopathy, prematurity retinopathy, retinal venous occlusion, metastasis of tumors SENJU PHARMACEUTICAL CO., LTD. (JP) 2003-04-22 US disclosed
EP-0771565-B1 Angiogenesis inhibitor SENJU PHARMA CO (JP) 2003-01-02 EP disclosed
US-6214800-B1 ANGIOGENESIS INHIBITORS SENJU PHARMACEUTICAL CO., LTD. (JP) 2001-04-10 US disclosed
US-6057290-A ADMINISTERING A CYSTEINE PROTEASE INHIBITOR TO A PATIENT FOR INHIBITING ANGIOGENESIS SENJU PHARMACEUTICAL CO., LTD. (JP) 2000-05-02 US disclosed
EP-0928786-A1 Angiogenesis inhibitor Senju Pharmaceutical Co., Ltd. (JP) 1999-07-14 EP disclosed
EP-0927716-A1 Angiogenesis inhibitor Senju Pharmaceutical Co., Ltd. (JP) 1999-07-07 EP disclosed
EP-0838460-A1 PIPERAZINE DERIVATIVES AND USE OF THE SAME Senju Pharmaceutical Co., Ltd. (JP) 1998-04-29 EP disclosed
EP-0771565-A2 Angiogenesis inhibitor Senju Pharmaceutical Co., Ltd. (JP) 1997-05-07 EP disclosed