SCHEMBL6981352

SCHEMBL6981352

COC(=O)CC(c1ccc(C)cc1)C1CCCC(=N)NC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.37
ALDH1A1 P00352 1/20 0.35
YAP1 P46937 1/20 0.35
TEAD4 Q15561 1/20 0.35
HTT P42858 1/20 0.34
HTR1E P28566 1/20 0.33
S1PR3 Q99500 1/20 0.33
HCRTR2 O43614 2/20 0.32
USP2 O75604 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974191 0.79 YAP1 (0.35) TSHRYAP1TEAD4
SCHEMBL6971316 0.74 RAB9A (0.38) TSHR
SCHEMBL10639565 0.73 ALDH1A1 (0.34) ALDH1A1HTT
SCHEMBL6977408 0.71 ALDH1A1 (0.55) ALDH1A1
SCHEMBL27797853 0.69 KMT2A (0.58) TSHR
SCHEMBL9413683 0.69 MEN1 (0.40) TSHRALDH1A1HTTHTR1ES1PR3
SCHEMBL435358 0.69 FFAR1 (0.48) ALDH1A1HTT
SCHEMBL13715266 0.69 FFAR1 (0.48) ALDH1A1HTT
SCHEMBL13715262 0.69 FFAR1 (0.48) ALDH1A1HTT
SCHEMBL9540511 0.68 SLC6A2 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP claimed