SCHEMBL6981483

SCHEMBL6981483

O=C(Nc1cccc2c1NCCC2)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.44
JAK2 O60674 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
KLK7 P49862 1/20 0.44
AKT1 P31749 1/20 0.42
ADRA2A P08913 1/20 0.41
PARP14 Q460N5 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
SLC13A5 Q86YT5 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.36
KDM4E B2RXH2 1/20 0.36
SLC18A3 Q16572 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5051442 0.81 SRC (0.47) SRCAKT1PARP14L3MBTL1KDM4E
SCHEMBL3316275 0.78 SRC (0.45) SRCAKT1SLC13A5ALDH1A1
SCHEMBL6984840 0.78 KDM4E (0.51) SRCTP53HTTAKT1L3MBTL1
SCHEMBL3728781 0.77 ALDH1A1 (0.58) ADRA2AL3MBTL1KDM4EMEN1KMT2A
SCHEMBL13903229 0.75 SRC (0.47) SRCMAPTHTTAKT1ADORA2A
SCHEMBL379494 0.75 SRC (0.47) SRCMAPTHTTAKT1ADRA2A
SCHEMBL6981450 0.75 AKT1 (0.52) MAPTHTTAKT1PARP14L3MBTL1
SCHEMBL18992141 0.73 JAK2 (0.42) JAK2TP53MAPTHTTKLK7
SCHEMBL28028253 0.72 SRC (0.45) SRCMAPTHTTAKT1ADRA2A
SCHEMBL16268278 0.72 CD44 (0.45) JAK2TP53MAPTHTTKLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed