SCHEMBL6984840

SCHEMBL6984840

O=C(Nc1cccc2c1NCCC2)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
SRC P12931 1/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
TP53 P04637 2/20 0.46
GAA P10253 1/20 0.46
NFKB1 P19838 1/20 0.46
HTT P42858 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 2/20 0.45
MDM4 O15151 1/20 0.45
HDAC3 O15379 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5051442 0.81 SRC (0.47) KDM4EL3MBTL1SRCNPC1RAB9A
SCHEMBL6981450 0.80 AKT1 (0.52) KDM4EL3MBTL1NPC1RAB9ACYP1A2
SCHEMBL6981483 0.78 SRC (0.44) KDM4EL3MBTL1SRCCYP1A2TP53
SCHEMBL6197534 0.77 CASP3 (0.50) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL28987534 0.77 L3MBTL1 (0.72) KDM4EL3MBTL1NPC1RAB9ATP53
SCHEMBL6054998 0.77 L3MBTL1 (0.76) KDM4EL3MBTL1POLBHPGDMEN1
SCHEMBL3316275 0.76 SRC (0.45) SRCPOLBMAPK1AKT1
SCHEMBL379494 0.75 SRC (0.47) KDM4EL3MBTL1SRCNPC1HTT
SCHEMBL28028253 0.72 SRC (0.45) KDM4ESRCNPC1HTTSMN1; SMN2
SCHEMBL8207031 0.72 L3MBTL1 (0.51) KDM4EL3MBTL1NPC1RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed