SCHEMBL6982020

SCHEMBL6982020

CN(C)C(=O)C=Cc1cccc(C2OCCO2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.39
IP6K1 Q92551 1/20 0.33
IP6K2 Q9UHH9 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
HDAC3 O15379 3/20 0.32
HDAC4 P56524 3/20 0.32
HDAC1 Q13547 3/20 0.32
HDAC7 Q8WUI4 3/20 0.32
HDAC2 Q92769 3/20 0.32
HDAC10 Q969S8 3/20 0.32
HDAC11 Q96DB2 3/20 0.32
HDAC8 Q9BY41 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
HDAC9 Q9UKV0 3/20 0.32
HDAC5 Q9UQL6 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4086910 0.74 CCR1 (0.35) KDM4EALDH1A1
SCHEMBL30147672 0.74 CCR1 (0.35) KDM4EALDH1A1
SCHEMBL12501420 0.73 NR4A2 (0.42) NR4A2IP6K1IP6K2CCNCCDK8
SCHEMBL6982026 0.71 RECQL (0.44) KDM4EMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL12501357 0.71 TGFBR1 (0.44) NR4A2CCNCCDK8KDM4EMAPT
SCHEMBL6975162 0.70 F2R (0.30)
SCHEMBL18095763 0.70 HTR1A (0.37)
SCHEMBL6983888 0.67 HTR1A (0.41) MEN1KMT2ASMN1; SMN2NPC1RAB9A
SCHEMBL24150010 0.67 KEAP1 (0.53) NR4A2CCNCCDK8KDM4EMAPT
SCHEMBL210591 0.67 KEAP1 (0.53) NR4A2CCNCCDK8KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946546-B1 PYRIDIN-2-YL-METHYLAMINE DERIVATIVES, METHOD OF PREPARING AND APPLICATION AS MEDICINE PF MEDICAMENT (FR) 2003-06-25 EP disclosed
US-6020345-A Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine PIERRE FABRE MEDICAMENT (FR) 2000-02-01 US disclosed