SCHEMBL6982169

SCHEMBL6982169

CON=C1C[C@H](C(=O)N2CCC(O)CC2)N(C(=O)c2ccc(-c3ccccc3)c(C)c2)C1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OXTR P30559 6/20 0.51
AVPR1A P37288 4/20 0.51
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
ROCK2 O75116 3/20 0.36
PDK2 Q15119 1/20 0.36
GABRA5 P31644 1/20 0.35
EPHX1 P07099 1/20 0.35
CYP46A1 Q9Y6A2 1/20 0.35
HPGD P15428 1/20 0.35
AVPR2 P30518 1/20 0.35
AVPR1B P47901 1/20 0.35
GRM5 P41594 1/20 0.34
L3MBTL3 Q96JM7 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4944058 0.89 AVPR1A (0.65) OXTRAVPR1AMEN1GAAMAPT
SCHEMBL4944054 0.89 AVPR1A (0.65) OXTRAVPR1AMEN1GAAMAPT
SCHEMBL4942034 0.88 OXTR (0.58) OXTRAVPR1AMEN1GAAMAPT
SCHEMBL4942028 0.88 OXTR (0.58) OXTRAVPR1AMEN1GAAMAPT
SCHEMBL5043513 0.87 AVPR1A (0.62) OXTRAVPR1AROCK2EPHX1AVPR2
SCHEMBL16550680 0.80 AVPR1A (0.78) OXTRAVPR1AROCK2PDK2EPHX1
SCHEMBL16550611 0.80 AVPR1A (0.78) OXTRAVPR1AROCK2PDK2EPHX1
SCHEMBL28754783 0.80 AVPR1A (0.78) OXTRAVPR1AROCK2PDK2EPHX1
SCHEMBL16550612 0.80 AVPR1A (0.78) OXTRAVPR1AROCK2PDK2EPHX1
SCHEMBL5474456 0.78 OXTR (0.61) OXTRAVPR1AMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268418-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001074769-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-11 WO disclosed