SCHEMBL5474456

SCHEMBL5474456

CON=C1C[C@@H](C(=O)NCCc2ccccc2)N(C(=O)c2ccc(-c3ccccc3)c(C)c2)C1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OXTR P30559 6/20 0.61
AVPR1A P37288 4/20 0.61
PTPN1 P18031 1/20 0.39
HDAC8 Q9BY41 3/20 0.38
PRSS1 P07477 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
ATM Q13315 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
FKBP1A P62942 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4942676 0.91 OXTR (0.73) OXTRAVPR1APTPN1HDAC8TAAR1
SCHEMBL5759282 0.91 OXTR (0.73) OXTRAVPR1APTPN1HDAC8TAAR1
SCHEMBL5043513 0.85 AVPR1A (0.62) OXTRAVPR1AROCK2
SCHEMBL7083271 0.85 OXTR (0.83) OXTRAVPR1APRSS1ROCK2ROCK1
SCHEMBL4945458 0.85 OXTR (0.83) OXTRAVPR1APRSS1ROCK2ROCK1
SCHEMBL4942915 0.81 AVPR1A (0.75) OXTRAVPR1A
SCHEMBL7086467 0.81 AVPR1A (0.75) OXTRAVPR1A
SCHEMBL7083946 0.81 AVPR1A (0.59) OXTRAVPR1A
SCHEMBL4939162 0.81 OXTR (0.73) OXTRAVPR1AHDAC8MEN1KMT2A
SCHEMBL4944329 0.81 OXTR (0.73) OXTRAVPR1AHDAC8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7211601-B2 Pharmaceutically active pyrrolidine derivatives APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2007-05-01 US disclosed