SCHEMBL6982528

SCHEMBL6982528

CCCCS(=O)(=O)Nc1cccc2c1N(C(=O)CCc1ccc(C(=N)N)cc1)CCC2

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 3/20 0.47
AVPR2 P30518 2/20 0.40
OXTR P30559 2/20 0.40
AVPR1A P37288 2/20 0.40
NR3C1 P04150 3/20 0.37
F2 P00734 2/20 0.37
PLG P00747 1/20 0.37
PRSS1 P07477 1/20 0.37
TPSAB1 Q15661 1/20 0.37
TPSD1 Q9BZJ3 1/20 0.37
TPSG1 Q9NRR2 1/20 0.37
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
ATM Q13315 1/20 0.35
F10 P00742 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981837 0.91 AVPR2 (0.39) AVPR2OXTRAVPR1ANR3C1ATM
SCHEMBL6984143 0.86 NR3C1 (0.37) AVPR2OXTRAVPR1ANR3C1ATM
SCHEMBL6982743 0.84 F2 (0.42) NR3C1F2PLGPRSS1TPSAB1
SCHEMBL6982524 0.82 NR3C1 (0.51) MRGPRX1AVPR2OXTRAVPR1ANR3C1
SCHEMBL6984822 0.82 SLC16A3 (0.40) MRGPRX1NR3C1F2PLGPRSS1
Hydrochloric Acid SCHEMBL6987687 0.81 NR3C1 (0.50) MRGPRX1AVPR2OXTRAVPR1ANR3C1
SCHEMBL6981750 0.81 AVPR2 (0.38) AVPR2OXTRAVPR1ANR3C1F2
SCHEMBL6982945 0.80 NR3C1 (0.36) AVPR2OXTRAVPR1ANR3C1ATM
SCHEMBL6986102 0.80 MAPT (0.41) F2PLGPRSS1TPSAB1TPSD1
SCHEMBL6982761 0.77 HDAC1 (0.35) NR3C1ATMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP claimed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO claimed
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed