SCHEMBL6981837

SCHEMBL6981837

CCCCS(=O)(=O)Nc1cccc2c1N(C(=O)CCc1ccc(CN)cc1)CCC2

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.39
OXTR P30559 2/20 0.39
AVPR1A P37288 2/20 0.39
NR3C1 P04150 2/20 0.37
MAPT P10636 3/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 1/20 0.37
ATM Q13315 1/20 0.36
GAA P10253 1/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 1/20 0.35
MEN1 O00255 1/20 0.35
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982528 0.91 MRGPRX1 (0.47) AVPR2OXTRAVPR1ANR3C1MAPT
SCHEMBL6984143 0.90 NR3C1 (0.37) AVPR2OXTRAVPR1ANR3C1MAPT
SCHEMBL6982945 0.84 NR3C1 (0.36) AVPR2OXTRAVPR1ANR3C1MAPT
SCHEMBL6984843 0.82 GAA (0.43) NR3C1GAAALDH1A1NPC1RAB9A
SCHEMBL6981833 0.81 NR3C1 (0.51) NR3C1MAPTLMNATP53GAA
SCHEMBL6982761 0.81 HDAC1 (0.35) NR3C1MAPTATMGAAALDH1A1
SCHEMBL6981764 0.80 METAP2 (0.42) MAPTLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL6982500 0.79 SLC16A3 (0.48) GAA
SCHEMBL6984787 0.76 ATM (0.48) MAPTTP53ATMALDH1A1NPC1
SCHEMBL6985566 0.76 PARP14 (0.40) NR3C1MAPTTP53ATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed