SCHEMBL6981750

SCHEMBL6981750

CCCCS(=O)(=O)N(CC(=O)O)c1cccc2c1N(C(=O)CCc1ccc(C(=N)N)cc1)CCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.38
OXTR P30559 2/20 0.38
AVPR1A P37288 2/20 0.38
ITGB3 P05106 7/20 0.38
ITGA2B P08514 7/20 0.38
NR3C1 P04150 2/20 0.37
F2 P00734 3/20 0.35
PLG P00747 1/20 0.35
PRSS1 P07477 1/20 0.35
TPSAB1 Q15661 1/20 0.35
TPSD1 Q9BZJ3 1/20 0.35
TPSG1 Q9NRR2 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
F10 P00742 2/20 0.33
PTGER4 P35408 1/20 0.33
PTGER2 P43116 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976368 0.88 ITGB3 (0.39) ITGB3ITGA2BF2PLGPRSS1
SCHEMBL6979635 0.85 ITGB3 (0.40) ITGB3ITGA2BF2PLGPRSS1
SCHEMBL6981742 0.84 NR3C1 (0.49) AVPR2OXTRAVPR1AITGB3ITGA2B
SCHEMBL6978680 0.82 KEAP1 (0.47) ITGB3ITGA2BF2PLGPRSS1
SCHEMBL6982528 0.81 MRGPRX1 (0.47) AVPR2OXTRAVPR1AITGB3ITGA2B
SCHEMBL6982999 0.80 ALDH1A1 (0.41) AVPR2OXTRAVPR1AITGB3ITGA2B
SCHEMBL6982234 0.79 TP53 (0.41) F2PLGPRSS1TPSAB1TPSD1
SCHEMBL6986115 0.79 ITGB3 (0.40) AVPR2OXTRAVPR1AITGB3ITGA2B
SCHEMBL6986000 0.78 NR3C1 (0.36) AVPR2OXTRAVPR1ANR3C1LMNA
SCHEMBL6984709 0.78 F2 (0.44) ITGB3ITGA2BF2PRSS1KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP claimed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP claimed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO claimed
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed