SCHEMBL6982617

SCHEMBL6982617

CC(C)(C)OC(=O)N1CCC(C(=O)N2CCCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)CC1

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.65
CNR1 P21554 1/20 0.65
NPSR1 Q6W5P4 1/20 0.64
STS P08842 2/20 0.60
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
HPGD P15428 1/20 0.56
TGM2 P21980 2/20 0.54
F13A1 P00488 1/20 0.54
TGM1 P22735 1/20 0.54
POLB P06746 1/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
TSHR P16473 1/20 0.53
ALDH1A1 P00352 1/20 0.53
PKM P14618 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979984 0.93 GAA (0.74) GAACNR1NPSR1STSNPC1
SCHEMBL6972262 0.90 NPC1 (0.56) GAANPC1RAB9AHPGDTGM2
SCHEMBL5736874 0.86 F10 (0.64) GAACNR1NPSR1STSTGM2
SCHEMBL5253160 0.86 POLB (0.70) GAACNR1STSTGM2F13A1
SCHEMBL6980123 0.85 LSS (0.60) GAACNR1HPGDTGM2F13A1
SCHEMBL6970591 0.82 GAA (0.72) GAACNR1NPSR1NPC1RAB9A
SCHEMBL7086266 0.82 ALDH1A1 (0.59) GAANPC1RAB9AHPGDTGM2
SCHEMBL1955697 0.81 ALDH1A1 (0.62) NPC1RAB9ATGM2F13A1TGM1
SCHEMBL6787216 0.80 KMT2A (0.65) GAARAB9AMEN1KMT2ATSHR
SCHEMBL14490210 0.80 TGM2 (0.59) TGM2F13A1TGM1ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925286-B1 SUBSTITUTED PYRIMIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ASTRAZENECA AB (SE) 2003-01-02 EP disclosed
US-6093718-A AN OXIDO-SQUALENE CYCLASE INHIBITOR, ANTICHOLESTEROL AGENT FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND LOWERING CHOLESTEROL LEVELS IN BLOOD PLASMA; TREATING HYPERCHOLESTEROLEMIA AND ATHEROSCLEROSIS ZENECA LIMITED (GB) 2000-07-25 US disclosed
EP-0925286-A1 SUBSTITUTED PYRIMIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ZENECA LIMITED (GB) 1999-06-30 EP disclosed
WO-1998006705-A1 SUBSTITUTED PYRIMIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ZENECA LIMITED (GB) 1998-02-19 WO disclosed