SCHEMBL6982875

SCHEMBL6982875

CCCC[C@H](NC(=O)NC(C)C(=O)O)C(=O)N(Cc1cccs1)Cc1cccs1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
CTSK P43235 3/20 0.43
GAA P10253 1/20 0.42
TRPM8 Q7Z2W7 3/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
FOLH1 Q04609 2/20 0.41
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6122567 0.90 CTSK (0.45) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL17388825 0.88 ALDH1A1 (0.43) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL6121971 0.87 CTSK (0.44) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL17388824 0.87 ALDH1A1 (0.45) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL6122977 0.87 TRPM8 (0.46) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL16762178 0.87 ALDH1A1 (0.46) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL16762075 0.87 ALDH1A1 (0.46) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL6123072 0.84 CTSK (0.46) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL6121764 0.84 CTSK (0.46) ALDH1A1CTSKGAATRPM8POLB
SCHEMBL6122227 0.84 CTSK (0.47) ALDH1A1CTSKGAATRPM8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071680-A4 N,N-DISUBSTITUTED AMIDES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS TEXAS BIOTECHNOLOGY CORP (US) 2003-03-05 EP disclosed
EP-1071680-A1 N,N-DISUBSTITUTED AMIDES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS TEXAS BIOTECHNOLOGY CORPORATION (US) 2001-01-31 EP disclosed
WO-1999052898-A1 N,N-DISUBSTITUTED AMIDES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS TEXAS BIOTECHNOLOGY CORPORATION (US) 1999-10-21 WO disclosed