SCHEMBL6984435

SCHEMBL6984435

COC(=O)[C@H](Cc1c[nH]c2ccc(O)cc12)NC(C)=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.58
NPSR1 Q6W5P4 5/20 0.56
BLM P54132 4/20 0.56
ALDH1A1 P00352 4/20 0.56
MAPT P10636 4/20 0.56
CYP1A2 P05177 3/20 0.56
CYP2D6 P10635 3/20 0.56
KDM4E B2RXH2 3/20 0.56
CYP3A4 P08684 3/20 0.56
SPR P35270 2/20 0.56
HPGD P15428 2/20 0.56
IDO1 P14902 1/20 0.56
NOTUM Q6P988 1/20 0.56
KMT2A Q03164 6/20 0.55
MEN1 O00255 4/20 0.55
HCRTR1 O43613 1/20 0.55
NFKB1 P19838 4/20 0.54
CYP2C9 P11712 3/20 0.54
CYP2C19 P33261 2/20 0.54
HTR1A P08908 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11734541 1.00 TACR1 (0.58) TACR1NPSR1BLMALDH1A1MAPT
SCHEMBL30359421 0.91 TACR1 (0.60) TACR1NPSR1BLMALDH1A1MAPT
SCHEMBL16626133 0.89 IL1RN (0.56) TACR1NPSR1BLMALDH1A1MAPT
SCHEMBL23501915 0.88 KMT2A (0.62) NPSR1BLMALDH1A1MAPTCYP1A2
SCHEMBL23501914 0.88 KMT2A (0.62) NPSR1BLMALDH1A1MAPTCYP1A2
SCHEMBL19252917 0.88 NPSR1 (0.63) NPSR1BLMALDH1A1MAPTCYP1A2
SCHEMBL3043368 0.88 NPSR1 (0.63) NPSR1BLMALDH1A1MAPTCYP1A2
SCHEMBL5115709 0.88 HTR2C (0.56) NPSR1BLMALDH1A1MAPTCYP1A2
SCHEMBL2857033 0.87 MTNR1A (0.61) TACR1BLMALDH1A1CYP1A2CYP2D6
SCHEMBL2857036 0.87 MTNR1A (0.61) TACR1BLMALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268422-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES Bayer Aktiengesellschaft (DE) 2003-01-02 EP disclosed
WO-2001070687-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-27 WO disclosed