SCHEMBL6984480

SCHEMBL6984480

Cc1cc(CCOc2cc[c]cc2)c2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.48
HTT P42858 2/20 0.48
PKM P14618 2/20 0.46
RXFP1 Q9HBX9 2/20 0.45
MAPK1 P28482 1/20 0.45
CYP1A2 P05177 1/20 0.44
MMP13 P45452 1/20 0.44
ADAM17 P78536 1/20 0.44
NCF1 P14598 2/20 0.42
ALDH1A1 P00352 4/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GLA P06280 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3974193 0.86 ADAM17 (0.57) SMN1; SMN2HTTMMP13ADAM17
SCHEMBL2528433 0.84 NPC1 (0.51) SMN1; SMN2HTTPKMRXFP1MAPK1
SCHEMBL6629881 0.81 SMN1; SMN2 (0.55) SMN1; SMN2HTTPKMRXFP1MAPK1
SCHEMBL6633283 0.79 SMN1; SMN2 (0.53) SMN1; SMN2HTTPKMRXFP1MAPK1
SCHEMBL6790022 0.78 NCF1 (0.60) SMN1; SMN2HTTCYP1A2NCF1ALDH1A1
SCHEMBL3967736 0.76 CYP1A2 (0.54) SMN1; SMN2HTTCYP1A2ADAM17NCF1
SCHEMBL6632245 0.75 ADAM17 (0.63) SMN1; SMN2HTTCYP1A2MMP13ADAM17
SCHEMBL7246568 0.73 LMNA (0.44) MMP13ADAM17ALDH1A1CASP1CASP7
SCHEMBL18535317 0.73 CYP1A2 (0.58) SMN1; SMN2HTTCYP1A2NCF1ALDH1A1
SCHEMBL3970289 0.72 SMN1; SMN2 (0.47) SMN1; SMN2HTTPKMRXFP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322627-A1 CYCLIC SULFONYL COMPOUNDS AS INHIBITORS OF METALLOPROTEASES Bristol-Myers Squibb Pharma Company (US) 2003-07-02 EP disclosed
WO-2002028846-A1 CYCLIC SULFONYL COMPOUNDS AS INHIBITORS OF METALLOPROTEASES DUPONT PHARMACEUTICALS COMPANY (US) 2002-04-11 WO disclosed