SCHEMBL6984495

SCHEMBL6984495

COc1cccc(C2CC(=O)C=C(C)N2)c1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
HTR2C P28335 2/20 0.44
LMNA P02545 1/20 0.43
MEN1 O00255 2/20 0.43
NPC1 O15118 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
CYP19A1 P11511 1/20 0.42
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981391 0.80 MAPT (0.43) LMNAMEN1KMT2AGAA
SCHEMBL6985757 0.80 MAPT (0.43) LMNAMEN1KMT2AGAA
SCHEMBL6978662 0.80 MAPT (0.43) LMNAMEN1KMT2AGAA
SCHEMBL6979945 0.79 BRD4 (0.45) LMNAMEN1KMT2A
SCHEMBL8538828 0.72 DDB1 (0.62) DDB1CRBNHTR2CMEN1NPC1
SCHEMBL6986386 0.72 CHRNB2 (0.46) LMNAMEN1KMT2AKDM4EALOX15
SCHEMBL7671819 0.72 DDB1 (0.54) DDB1CRBNHTR2CMEN1NPC1
SCHEMBL29144920 0.71 CYP19A1 (0.50) DDB1CRBNHTR2CLMNAMEN1
SCHEMBL30688767 0.71 CYP19A1 (0.50) DDB1CRBNHTR2CLMNAMEN1
SCHEMBL29144948 0.71 CYP19A1 (0.50) DDB1CRBNHTR2CLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1050530-B1 1-Aza-2-alkyl-6-aryl-cycloalkanes usefull as memory enhancers SERVIER LAB (FR) 2003-10-22 EP disclosed
US-6451789-B1 CENTRAL NERVOUS SYSTEM DISORDERS; COGNITION ACTIVATORS LES LABORTOIRES SERVIER (FR) 2002-09-17 US disclosed
US-20020042413-A1 1-aza-2-alkyl-6-aryl-cycloalkanes RAULT SYLVAIN (FR) 2002-04-11 US disclosed
US-6323222-B1 COGNITION ACTIVATORS, ALZHEIMER*S DISEASE AND ENZYME INHIBITORS ADIR ET COMPAGNIE (FR) 2001-11-27 US disclosed
EP-1050530-A1 1-Aza-2-alkyl-6-aryl-cycloalkanes usefull as memory enhancers ADIR ET COMPAGNIE (FR) 2000-11-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020042413-A1 1-aza-2-alkyl-6-aryl-cycloalkanes SULT2A1, GRIN2A, NR3C1 DDB1 1816/4885CRBN 1839/4885HTR2C 137/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.