SCHEMBL6984553

SCHEMBL6984553

N#Cc1ccc(C=CC(=O)N2CCCc3cc(NS(=O)(=O)c4ccccc4)ccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 8/20 0.56
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
TP53 P04637 3/20 0.48
MAPT P10636 3/20 0.48
LMNA P02545 2/20 0.47
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
PKM P14618 1/20 0.46
DRD2 P14416 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
DRD3 P35462 1/20 0.46
HTR6 P50406 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984550 1.00 NR3C1 (0.56) NR3C1ALDH1A1MEN1RAB9AKMT2A
Hydrochloric Acid SCHEMBL6984889 0.85 NR3C1 (0.56) NR3C1ALDH1A1MEN1RAB9AKMT2A
SCHEMBL6985366 0.84 NR3C1 (0.66) NR3C1ALDH1A1RAB9ATP53MAPT
SCHEMBL6984554 0.82 ALDH1A1 (0.44) NR3C1ALDH1A1MEN1RAB9AKMT2A
SCHEMBL6983044 0.80 NR3C1 (0.58) NR3C1TP53MAPTLMNAPKM
SCHEMBL6980538 0.80 NR3C1 (0.56) NR3C1ALDH1A1TP53MAPTLMNA
SCHEMBL6985317 0.80 NR3C1 (0.58) NR3C1MEN1KMT2ATP53MAPT
SCHEMBL6981758 0.79 NR3C1 (0.56) NR3C1TP53MAPTLMNAPKM
SCHEMBL6977969 0.79 NR3C1 (0.56) NR3C1ALDH1A1MEN1KMT2ATP53
SCHEMBL6982976 0.78 NR3C1 (0.54) NR3C1TP53MAPTLMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed