SCHEMBL6984554

SCHEMBL6984554

N#Cc1ccc(C=CC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccccc4)c32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
RAB9A P51151 1/20 0.44
LMNA P02545 5/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.42
NR3C1 P04150 2/20 0.40
AR P10275 1/20 0.40
P4HB P07237 1/20 0.40
MAPT P10636 3/20 0.39
PKM P14618 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HDAC3 O15379 2/20 0.39
HDAC4 P56524 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC7 Q8WUI4 2/20 0.39
HDAC2 Q92769 2/20 0.39
HDAC10 Q969S8 2/20 0.39
HDAC11 Q96DB2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985371 0.84 NR3C1 (0.44) ALDH1A1LMNAGAANR3C1AR
SCHEMBL6984550 0.82 NR3C1 (0.56) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL6984553 0.82 NR3C1 (0.56) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL6983048 0.80 NAMPT (0.41) ALDH1A1MEN1KMT2ALMNANR3C1
SCHEMBL6985322 0.80 GAA (0.41) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL6980541 0.80 HSD17B10 (0.48) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL6982980 0.78 PKM (0.39) ALDH1A1MEN1KMT2ALMNAHPGD
SCHEMBL7406048 0.78 EEF2K (0.39) ALDH1A1MEN1KMT2ALMNAHPGD
SCHEMBL6981761 0.78 LIMK2 (0.40) ALDH1A1MEN1KMT2ALMNAHPGD
SCHEMBL6976883 0.78 NR3C1 (0.38) ALDH1A1MEN1KMT2ARAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed