SCHEMBL6984610

SCHEMBL6984610

CC(C)(C)NC(=O)N1CCN(C(=O)SC(=O)c2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
GAA P10253 3/20 0.43
LMNA P02545 1/20 0.43
CNR1 P21554 3/20 0.43
CNR2 P34972 2/20 0.43
CSNK1E P49674 5/20 0.42
CSNK1D P48730 1/20 0.41
RBP4 P02753 1/20 0.40
TSHR P16473 1/20 0.40
P2RY12 Q9H244 1/20 0.40
RORC P51449 1/20 0.39
CYP2C9 P11712 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987678 0.81 CYP3A4 (0.47) GAACNR1TSHRCYP2C9SMN1; SMN2
SCHEMBL4677423 0.80 KDM4E (0.56) GAACYP2C9SMN1; SMN2
Hydrochloric Acid SCHEMBL4681386 0.80 CYP3A4 (0.46) GAACNR1TSHRCYP2C9SMN1; SMN2
Hydrochloric Acid SCHEMBL6990408 0.80 KMT2A (0.51) RAB9AGAACNR1CNR2RBP4
Hydrochloric Acid SCHEMBL6993204 0.79 POLB (0.56) GAACYP2C9
SCHEMBL6983830 0.77 GPR139 (0.50) NPC1LMNAP2RY12
SCHEMBL6987979 0.77 KDM4E (0.59) LMNASMN1; SMN2
SCHEMBL6987336 0.76 CNR1 (0.59) GAACNR1CNR2SMN1; SMN2
Hydrochloric Acid SCHEMBL6988112 0.76 GPR139 (0.49) NPC1LMNAP2RY12
Hydrochloric Acid SCHEMBL6991722 0.76 KDM4E (0.58) LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343775-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-09-17 EP disclosed
WO-2002048124-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-20 WO disclosed