SCHEMBL6987979

SCHEMBL6987979

O=C(SC(=O)N1CCN(C(=O)NCc2ccccc2)CC1)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.59
HRH3 Q9Y5N1 1/20 0.55
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
NPSR1 Q6W5P4 1/20 0.54
TPSAB1 Q15661 2/20 0.54
TP53 P04637 1/20 0.54
F2 P00734 1/20 0.52
PRSS1 P07477 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
LMNA P02545 1/20 0.51
HTT P42858 1/20 0.51
RECQL P46063 1/20 0.51
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48
TUBB3 Q13509 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6991722 0.99 KDM4E (0.58) KDM4EHRH3MEN1KMT2ANPSR1
SCHEMBL6992011 0.88 PKM (0.59) KDM4EHRH3MEN1KMT2A
SCHEMBL6987380 0.88 CTDSP1 (0.57) KDM4EHRH3MEN1KMT2ANPSR1
Hydrochloric Acid SCHEMBL6987696 0.87 CTDSP1 (0.56) KDM4EHRH3MEN1KMT2ANPSR1
Hydrochloric Acid SCHEMBL6989166 0.87 PKM (0.58) KDM4EHRH3MEN1KMT2A
Hydrochloric Acid SCHEMBL6990408 0.84 KMT2A (0.51) KDM4EMEN1KMT2ASMN1; SMN2HTT
SCHEMBL6991815 0.84 ALDH1A1 (0.52) KDM4EMEN1KMT2ALMNAHTT
Hydrochloric Acid SCHEMBL6990747 0.83 ALDH1A1 (0.51) KDM4EMEN1KMT2ALMNAHTT
SCHEMBL4677795 0.82 LMNA (0.45) KDM4EMEN1KMT2ALMNAALDH1A1
Hydrochloric Acid SCHEMBL6988072 0.82 EPHX2 (0.42) KDM4EMEN1KMT2ATPSAB1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343775-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-09-17 EP claimed
WO-2002048124-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-20 WO claimed
EP-1343775-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-09-17 EP disclosed
WO-2002048124-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-20 WO disclosed