SCHEMBL6984795

SCHEMBL6984795

CC(C)(C)OC(=O)COc1ccc2oc(C(=O)O)cc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 4/20 0.55
LMNA P02545 3/20 0.50
TP53 P04637 1/20 0.50
HPGD P15428 4/20 0.48
POLB P06746 3/20 0.48
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.48
BLM P54132 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
THRA P10827 1/20 0.48
THRB P10828 1/20 0.48
PIM2 Q9P1W9 1/20 0.46
MAPT P10636 3/20 0.45
CYP2C19 P33261 2/20 0.45
CYP2C9 P11712 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
FLT3 P36888 1/20 0.45
CA2 P00918 2/20 0.42
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL541866 0.88 PIM1 (0.53) PIM1LMNATP53HPGDPOLB
SCHEMBL6984136 0.84 POLB (0.51) PIM1LMNAHPGDPOLBALDH1A1
SCHEMBL26109666 0.83 PIM1 (0.58) PIM1LMNATP53HPGDPOLB
SCHEMBL13765283 0.81 CYP2A6 (0.43) LMNAHPGDPOLBALDH1A1MEN1
SCHEMBL12529923 0.80 CA12 (0.54) PIM1LMNATP53HPGDPOLB
SCHEMBL30540812 0.80 CA12 (0.54) PIM1LMNATP53HPGDPOLB
SCHEMBL10066356 0.80 PIM1 (0.50) PIM1LMNATP53HPGDPOLB
SCHEMBL5866928 0.80 ALDH1A1 (0.68) PIM1LMNATP53HPGDPOLB
SCHEMBL18591899 0.78 PIM1 (0.58) PIM1LMNATP53HPGDPOLB
SCHEMBL9990974 0.78 PIM1 (0.58) PIM1LMNATP53HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed