SCHEMBL10066356

SCHEMBL10066356

CC(C)(C)OC(=O)PCCOc1ccc2oc(C(=O)O)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 5/20 0.50
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
BLM P54132 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
PIM2 Q9P1W9 2/20 0.41
FLT3 P36888 1/20 0.41
CA2 P00918 2/20 0.38
TAS1R3 Q7RTX0 3/20 0.38
TAS1R1 Q7RTX1 3/20 0.38
PTGER4 P35408 2/20 0.38
MAOB P27338 2/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL541866 0.83 PIM1 (0.53) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL6984795 0.80 PIM1 (0.55) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL30540812 0.80 CA12 (0.54) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL12529923 0.80 CA12 (0.54) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL9990974 0.78 PIM1 (0.58) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL18591899 0.78 PIM1 (0.58) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL6414543 0.77 LMNA (0.62) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL5866928 0.75 ALDH1A1 (0.68) PIM1LMNATP53ALDH1A1HPGD
SCHEMBL4765626 0.75 DRD2 (0.52) PIM1CA2MAOBCA12CA1
SCHEMBL11457413 0.75 PIM1 (0.54) PIM1LMNATP53ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948242-B9 CYTOTOXIC COMPOUNDS MEDAREX INC (US) 2012-02-08 EP disclosed
EP-1948242-B1 CYTOTOXIC COMPOUNDS MEDAREX INC (US) 2011-09-14 EP disclosed