SCHEMBL6985351

SCHEMBL6985351

CC1CC(C)CN(C(=O)c2ccc3c(c2)CCCN3C(=O)CCc2ccc(C#N)cc2)C1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
TP53 P04637 1/20 0.44
KDM1A O60341 11/20 0.42
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410530 0.90 TP53 (0.45) ALDH1A1TP53KDM1AHDAC1HDAC8
SCHEMBL6981826 0.87 PDK1 (0.52) ALDH1A1TP53KDM1AHDAC1HDAC8
Hydrochloric Acid SCHEMBL7958653 0.87 F2 (0.42) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL6987041 0.84 CDK1 (0.45) ALDH1A1TP53HDAC1HDAC8HDAC6
SCHEMBL6985353 0.81 ALDH1A1 (0.46) ALDH1A1
SCHEMBL6985246 0.81 TP53 (0.51) ALDH1A1TP53HDAC1HDAC8HDAC6
SCHEMBL7948815 0.81 TP53 (0.42) ALDH1A1TP53HDAC1HDAC8HDAC6
SCHEMBL6986538 0.80 TP53 (0.49) ALDH1A1TP53HDAC1HDAC8HDAC6
SCHEMBL6977395 0.79 TP53 (0.46) ALDH1A1TP53HDAC1HDAC8HDAC6
SCHEMBL6985141 0.79 AVPR2 (0.47) ALDH1A1TP53KDM1AHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed