SCHEMBL6985802

SCHEMBL6985802

Cc1cc(Br)nc(CO)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.37
NOS2 P35228 10/20 0.36
NOS3 P29474 6/20 0.36
NOS1 P29475 6/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CCR1 P32246 1/20 0.32
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12161257 0.84 NOS2 (0.43) S1PR2NOS2NOS3NOS1ALDH1A1
Hydrochloric Acid SCHEMBL18640616 0.81 NOS2 (0.41) S1PR2NOS2NOS3NOS1CCR1
SCHEMBL18611531 0.80 NOS2 (0.57) NOS2NOS3NOS1
SCHEMBL13729089 0.78 CCR1 (0.32) CCR1
SCHEMBL18640608 0.78 S1PR2 (0.37) S1PR2NOS2NOS3NOS1CCR1
SCHEMBL667378 0.77 NOS2 (0.44) S1PR2NOS2NOS3NOS1KDM4E
SCHEMBL10367813 0.76 S1PR2 (0.38) S1PR2NOS2NOS3NOS1KDM4E
SCHEMBL20072591 0.76 NOS2 (0.57) S1PR2NOS2NOS3NOS1CCR1
SCHEMBL1821173 0.75
SCHEMBL20063090 0.75 NOS2 (0.52) S1PR2NOS2NOS3NOS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946546-B1 PYRIDIN-2-YL-METHYLAMINE DERIVATIVES, METHOD OF PREPARING AND APPLICATION AS MEDICINE PF MEDICAMENT (FR) 2003-06-25 EP disclosed
US-6020345-A Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine PIERRE FABRE MEDICAMENT (FR) 2000-02-01 US disclosed
EP-0946546-A1 PYRIDIN-2-YL-METHYLAMINE DERIVATIVES, METHOD OF PREPARING AND APPLICATION AS MEDICINE PIERRE FABRE MEDICAMENT (FR) 1999-10-06 EP disclosed
WO-1998022459-A1 PYRIDIN-2-YL-METHYLAMINE DERIVATIVES, METHOD OF PREPARING AND APPLICATION AS MEDICINE PIERRE FABRE MEDICAMENT (FR) 1998-05-28 WO disclosed