SCHEMBL20063090

SCHEMBL20063090

Cc1cc(CO)nc(C(C)C)c1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 0.52
NOS3 P29474 6/20 0.52
NOS1 P29475 6/20 0.52
S1PR2 O95136 1/20 0.35
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CCR1 P32246 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12161257 0.80 NOS2 (0.43) NOS2NOS3NOS1S1PR2ALDH1A1
SCHEMBL20063089 0.80 ACHE (0.38) NOS2NOS3NOS1CCR1
SCHEMBL15274618 0.80 NOS2 (0.38) NOS2NOS3NOS1CCR1
SCHEMBL4049194 0.80 NOS3 (0.34) NOS2NOS3NOS1CCR1
Hydrochloric Acid SCHEMBL18640616 0.78 NOS2 (0.41) NOS2NOS3NOS1S1PR2CCR1
SCHEMBL6662711 0.78 NOS2 (0.70) NOS2NOS3NOS1ALDH1A1
SCHEMBL12250770 0.76 NOS2 (0.61) NOS2NOS3NOS1S1PR2KDM4E
SCHEMBL21211968 0.76 NOS1 (0.53) NOS2NOS3NOS1
SCHEMBL6985802 0.75 S1PR2 (0.37) NOS2NOS3NOS1S1PR2KDM4E
SCHEMBL3506786 0.74 HRH3 (0.42) NOS2NOS3NOS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180105508-A1 INHIBITORS OF PHOSPHOGLYCERATE DEHYDROGENASE (PHGDH) AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2018-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180105508-A1 INHIBITORS OF PHOSPHOGLYCERATE DEHYDROGENASE (PHGDH) AND USES THEREOF PHGDH, PGD, PGK1 NOS2 2680/4885NOS3 2532/4885NOS1 2516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.