SCHEMBL6985909

SCHEMBL6985909

CC(C)C[C@@](Cc1ccccc1)(C(=O)O)[C@H](CCOS(C)(=O)=O)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
PSMB5 P28074 2/20 0.34
REN P00797 1/20 0.34
CTSS P25774 3/20 0.33
CTSK P43235 2/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
SYK P43405 1/20 0.33
MMP1 P03956 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
BACE1 P56817 3/20 0.32
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981175 0.85 CTSS (0.37) RENCTSSCTSKCTSLCTSB
SCHEMBL6988956 0.76 HTR2A (0.36) CTSSCTSKCTSLCTSBMMP1
SCHEMBL14713246 0.72 SMN1; SMN2 (0.46) MAPT
SCHEMBL6985583 0.72 REN (0.37) RENCTSL
SCHEMBL6985902 0.72 POLB (0.41) PSMB5CTSKSYKMAPT
SCHEMBL2856553 0.69 PPARA (0.51) CTSSCTSKCTSLCTSBSYK
SCHEMBL6775947 0.69 PPARA (0.51) CTSSCTSKCTSLCTSBSYK
SCHEMBL6985905 0.69 CTSS (0.36) CA12CA1CA7CA14REN
SCHEMBL5682158 0.68 PSMB5 (0.40) PSMB5CTSKSYKMAPT
SCHEMBL5677953 0.68 PSMB5 (0.40) PSMB5CTSKSYKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed