SCHEMBL6985905

SCHEMBL6985905

CC(CCc1ccccc1)CC(C(=O)O)[C@H](CCOS(C)(=O)=O)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
PRSS1 P07477 2/20 0.34
CTSG P08311 2/20 0.34
CTRB1 P17538 2/20 0.34
CMA1 P23946 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CYP24A1 Q07973 1/20 0.34
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34
NPR3 P17342 1/20 0.34
REN P00797 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981171 0.85 CTSS (0.40) CTSSCTSKITGA4ITGB7PRSS1
SCHEMBL6984941 0.81 CTSS (0.39) CTSSCTSKITGA4ITGB7PRSS1
SCHEMBL6985902 0.80 POLB (0.41) CTSK
SCHEMBL6988954 0.77 ALDH1A1 (0.41) CTSSCTSKITGA4ITGB7CYP24A1
SCHEMBL6659520 0.75 MMP3 (0.45) CTSSCTSKMMP1MMP3MMP9
SCHEMBL6943292 0.75 MMP3 (0.45) CTSSCTSKMMP1MMP3MMP9
SCHEMBL6987281 0.75 MMP3 (0.45) CTSSCTSKMMP1MMP3MMP9
SCHEMBL6659518 0.75 MMP3 (0.45) CTSSCTSKMMP1MMP3MMP9
SCHEMBL6943287 0.75 MMP3 (0.45) CTSSCTSKMMP1MMP3MMP9
SCHEMBL5682158 0.74 PSMB5 (0.40) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed