SCHEMBL6986423

SCHEMBL6986423

Cc1[nH]c2ccccc2c1-c1ccc(N)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.65
CYP1A2 P05177 2/20 0.54
CYP2C9 P11712 2/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
AHR P35869 1/20 0.50
LMNA P02545 2/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ESR1 P03372 4/20 0.47
ESR2 Q92731 4/20 0.47
PTGS2 P35354 3/20 0.47
CCR6 P51684 1/20 0.46
HKDC1 Q2TB90 1/20 0.46
ACHE P22303 1/20 0.46
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16169793 0.85 IMPDH2 (0.69) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL17383846 0.85 IMPDH2 (0.73) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL27701196 0.82 IMPDH2 (0.65) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL4607984 0.82 ESR1 (0.69) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL8722197 0.82 IMPDH2 (0.65) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL27566954 0.79 PTGS2 (0.62) IMPDH2MEN1KMT2AAHRLMNA
SCHEMBL8722153 0.79 IMPDH2 (0.65) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL31060312 0.79 IMPDH2 (1.00) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL28643376 0.78 IMPDH2 (0.59) IMPDH2CYP1A2CYP2C9MEN1KMT2A
SCHEMBL14023506 0.78 KMT2A (0.52) IMPDH2CYP1A2CYP2C9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303508-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2003-04-23 EP disclosed
WO-2002006273-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-01-24 WO disclosed