SCHEMBL6986658

SCHEMBL6986658

CC1CCC(c2cccc(NC(=O)Nc3ccc4ncccc4c3)c2)(N2CCN(c3ccccc3)CC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 2/20 0.51
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
NAMPT P43490 3/20 0.44
TRPV1 Q8NER1 2/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
CDK5 Q00535 1/20 0.42
PABPC1 P11940 1/20 0.42
HTR1A P08908 4/20 0.41
DRD2 P14416 3/20 0.41
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2A P28223 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6990046 0.99 NPY1R (0.50) NPY1RMEN1NPC1POLBMAPT
SCHEMBL6990201 0.91 NPY1R (0.51) NPY1RNPC1POLBMAPTNAMPT
Hydrochloric Acid SCHEMBL6992260 0.90 NPY1R (0.51) NPY1RNPC1POLBMAPTNAMPT
Hydrochloric Acid SCHEMBL6990944 0.88 NPY1R (0.55) NPY1RMEN1NPC1POLBMAPT
SCHEMBL7090848 0.86 HTR1A (0.55) NPY1RMEN1NPC1POLBMAPT
Hydrochloric Acid SCHEMBL6993221 0.86 HTR1A (0.54) NPY1RMEN1NPC1POLBMAPT
SCHEMBL7091275 0.85 HTR1A (0.54) NPY1RMEN1NPC1MAPTKMT2A
SCHEMBL7088429 0.85 TRPV1 (0.46) NPY1RMEN1NPC1POLBMAPT
Hydrochloric Acid SCHEMBL6989924 0.85 TRPV1 (0.46) NPY1RMEN1NPC1POLBMAPT
Hydrochloric Acid SCHEMBL6990799 0.85 HTR1A (0.54) NPY1RMEN1NPC1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915859-B1 CERTAIN SUBSTITUTED BENZYLAMINE DERIVATIVES; A NEW CLASS OF NEUROPEPTIDE Y1 SPECIFIC LIGANDS NEUROGEN CORP (US) 2003-01-02 EP claimed
EP-0915859-B1 CERTAIN SUBSTITUTED BENZYLAMINE DERIVATIVES; A NEW CLASS OF NEUROPEPTIDE Y1 SPECIFIC LIGANDS NEUROGEN CORP (US) 2003-01-02 EP disclosed
EP-0915859-A1 CERTAIN SUBSTITUTED BENZYLAMINE DERIVATIVES; A NEW CLASS OF NEUROPEPTIDE Y1 SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 1999-05-19 EP disclosed
WO-1998003492-A1 CERTAIN SUBSTITUTED BENZYLAMINE DERIVATIVES; A NEW CLASS OF NEUROPEPTIDE Y1 SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 1998-01-29 WO disclosed