SCHEMBL6987115

SCHEMBL6987115

CC(C)[Si](Oc1ccc(C(Br)(C=O)c2ccncc2)cc1)(C(C)C)C(C)C

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
CYP3A4 P08684 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988060 0.85 CYP3A4 (0.41) LMNACYP3A4ALDH1A1TDP1CYP1A2
SCHEMBL10958010 0.79 CYP1A2 (0.50) LMNACYP3A4ALDH1A1TDP1KDM4E
SCHEMBL6988582 0.74 CYP17A1 (0.35) LMNACYP3A4ALDH1A1TP53MAPK1
SCHEMBL6990626 0.70 CYP19A1 (0.33)
SCHEMBL3697133 0.70 ALDH1A3 (0.57) LMNAALDH1A1KDM4EHPGDSMN1; SMN2
Bromide SCHEMBL8081397 0.70 KIF11 (0.52) ALDH1A1CYP1A2RAB9A
SCHEMBL6991066 0.69 CYP19A1 (0.35) NPC1HPGDRAB9ASMN1; SMN2
Bromide SCHEMBL8121179 0.68 USP2 (0.55) RAB9A
SCHEMBL6179860 0.67 SMN1; SMN2 (0.36) LMNACYP3A4ALDH1A1TP53HPGD
SCHEMBL481885 0.67 MAPT (0.37) LMNAALDH1A1MAPK1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1328522-A2 ESTROGEN RECEPTOR MODULATORS Merck & Co., Inc. (US) 2003-07-23 EP disclosed
WO-2002032373-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO., INC. (US) 2002-04-25 WO disclosed