SCHEMBL6987236

SCHEMBL6987236

Cc1ccc(C)c2c(OCCN)noc12

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.35
CHEK1 O14757 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PRKCH P24723 1/20 0.32
PRKCE Q02156 1/20 0.32
PRKCQ Q04759 1/20 0.32
PRKCD Q05655 1/20 0.32
FAAH O00519 1/20 0.32
MGLL Q99685 1/20 0.32
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29416851 1.00 CYP17A1 (0.35) CYP17A1CHEK1TAAR1KDM4EPRKCH
Hydrochloric Acid SCHEMBL6992724 0.98 KDM4E (0.35) CYP17A1CHEK1TAAR1KDM4EPRKCH
SCHEMBL6989532 0.91 IDO1 (0.33) CYP17A1CHEK1
Hydrochloric Acid SCHEMBL6989390 0.90 IDO1 (0.33) CYP17A1CHEK1KDM4E
SCHEMBL29973407 0.88 CHEK1 (0.35) CYP17A1CHEK1KMT2A
Hydrochloric Acid SCHEMBL6990286 0.87 CYP17A1 (0.33) CYP17A1CHEK1KDM4EKMT2A
Hydrochloric Acid SCHEMBL6994412 0.87 CYP17A1 (0.31) CYP17A1KDM4E
Hydrochloric Acid SCHEMBL6995997 0.86 CHEK1 (0.34) CYP17A1CHEK1KDM4EKMT2A
Hydrochloric Acid SCHEMBL6990622 0.85 MBOAT4 (0.34) CYP17A1
Hydrochloric Acid SCHEMBL6993592 0.84 MKNK1 (0.36) KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779281-B1 ISOXAZOLES SANKYO CO (JP) 2003-10-29 EP claimed
US-6096771-A ISOXAZOLE DERIVATIVES EXHIBITING EXCELLENT TYPE B AND TYPE A MONOAMINE OXIDASE INHIBITORY ACTIVITIES, THEREFORE USEFUL FOR PREVENTING PARKINSON'S DISEASE, DEPRESSION AND ALZHEIMER'S DISEASE SANKYO COMPANY, LIMITED (JP) 2000-08-01 US claimed
CN-1162957-A Isoxazole derivatives SANKYO CO (JP) 1997-10-22 CN disclosed