SCHEMBL6989532

SCHEMBL6989532

Cc1ccc(F)c2c(OCCN)noc12

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.33
CYP17A1 P05093 2/20 0.33
CHEK1 O14757 1/20 0.33
KIT P10721 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6989390 0.99 IDO1 (0.33) IDO1CYP17A1CHEK1KITKDR
SCHEMBL29416851 0.91 CYP17A1 (0.35) CYP17A1CHEK1
SCHEMBL6987236 0.91 CYP17A1 (0.35) CYP17A1CHEK1
Hydrochloric Acid SCHEMBL6992724 0.89 KDM4E (0.35) CYP17A1CHEK1
Hydrochloric Acid SCHEMBL6994412 0.82 CYP17A1 (0.31) CYP17A1
Hydrochloric Acid SCHEMBL6990286 0.82 CYP17A1 (0.33) CYP17A1CHEK1KITKDRFLT3
Hydrochloric Acid SCHEMBL6990622 0.80 MBOAT4 (0.34) CYP17A1
SCHEMBL29973407 0.79 CHEK1 (0.35) CYP17A1CHEK1
Hydrochloric Acid SCHEMBL6993592 0.79 MKNK1 (0.36)
SCHEMBL8201516 0.78 FAAH (0.34) IDO1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779281-B1 ISOXAZOLES SANKYO CO (JP) 2003-10-29 EP claimed
US-6096771-A ISOXAZOLE DERIVATIVES EXHIBITING EXCELLENT TYPE B AND TYPE A MONOAMINE OXIDASE INHIBITORY ACTIVITIES, THEREFORE USEFUL FOR PREVENTING PARKINSON'S DISEASE, DEPRESSION AND ALZHEIMER'S DISEASE SANKYO COMPANY, LIMITED (JP) 2000-08-01 US claimed