SCHEMBL6987369

SCHEMBL6987369

COc1ccccc1-c1ccc(C(=O)N2CCc3nc(C)[nH]c3-c3ccccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 1/20 0.47
AVPR1A P37288 1/20 0.47
CDK4 P11802 1/20 0.46
CCND1 P24385 1/20 0.46
ROCK2 O75116 1/20 0.46
HTR1D P28221 4/20 0.45
HTR1B P28222 4/20 0.45
FFAR2 O15552 4/20 0.43
DHODH Q02127 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPK14 Q16539 1/20 0.42
PDCD1 Q15116 2/20 0.42
CD274 Q9NZQ7 2/20 0.42
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
GHSR Q92847 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6990553 0.99 AVPR2 (0.47) AVPR2AVPR1ACDK4CCND1ROCK2
SCHEMBL1495892 0.86 AVPR2 (0.50) AVPR2AVPR1ARAB9ASMN1; SMN2PDCD1
SCHEMBL7019597 0.84 ROCK2 (0.46) AVPR2AVPR1AROCK2DHODHRAB9A
SCHEMBL7019311 0.84 ROCK2 (0.46) AVPR2AVPR1AROCK2RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL6986424 0.84 AVPR2 (0.58) AVPR2AVPR1ARAB9AALDH1A1
Hydrochloric Acid SCHEMBL6994121 0.82 AVPR2 (0.46) AVPR2AVPR1ASMN1; SMN2MEN1KMT2A
SCHEMBL6993115 0.81 AVPR2 (0.45) AVPR2AVPR1ARAB9ASMN1; SMN2KMT2A
SCHEMBL6991735 0.81 HTR1D (0.45) CDK4CCND1ROCK2HTR1DHTR1B
SCHEMBL1821311 0.80 AVPR2 (0.56) AVPR2AVPR1APDCD1CD274POLB
SCHEMBL6987926 0.79 AVPR2 (0.68) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709386-B1 FUSED BENZAZEPINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMA CO LTD (JP) 2003-05-07 EP disclosed
EP-1097920-A1 Intermediate for condensed benzazepine derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2001-05-09 EP disclosed
EP-0709386-A1 FUSED BENZAZEPINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-05-01 EP disclosed