SCHEMBL6991735

SCHEMBL6991735

COc1ccccc1-c1ccc(C(=O)N2CCc3nc(C)oc3-c3ccccc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 4/20 0.45
HTR1B P28222 4/20 0.45
ROCK2 O75116 1/20 0.44
FFAR2 O15552 6/20 0.43
PDCD1 Q15116 3/20 0.43
CD274 Q9NZQ7 3/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
TP53 P04637 1/20 0.42
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1495876 0.86 ALDH1A1 (0.49) PDCD1CD274RAB9ASMN1; SMN2TP53
SCHEMBL6987369 0.81 AVPR2 (0.47) HTR1DHTR1BROCK2FFAR2PDCD1
Hydrochloric Acid SCHEMBL6990553 0.80 AVPR2 (0.47) HTR1DHTR1BROCK2FFAR2PDCD1
SCHEMBL6993535 0.79 AVPR2 (0.59)
SCHEMBL6619403 0.79 AVPR2 (0.65)
SCHEMBL2703870 0.78 PDCD1 (0.42) PDCD1CD274RAB9ASMN1; SMN2ALDH1A1
SCHEMBL2616280 0.77 PDCD1 (0.49) PDCD1CD274RAB9AMEN1KMT2A
Hydrochloric Acid SCHEMBL2129494 0.76 PDCD1 (0.48) PDCD1CD274RAB9AMEN1KMT2A
SCHEMBL6988182 0.76 ALDH1A1 (0.54) HTR1DHTR1BFFAR2RAB9ASMN1; SMN2
SCHEMBL27789716 0.75 PDCD1 (0.44) PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709386-B1 FUSED BENZAZEPINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMA CO LTD (JP) 2003-05-07 EP disclosed
EP-1097920-A1 Intermediate for condensed benzazepine derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2001-05-09 EP disclosed
EP-0709386-A1 FUSED BENZAZEPINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-05-01 EP disclosed