SCHEMBL6987648

SCHEMBL6987648

Cc1nn(C(CCCc2ccccc2)C(C)O)c2nc(Cc3ccccc3)[nH]c(=O)c12

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 5/20 0.47
CCNE1 P24864 7/20 0.41
CDK2 P24941 7/20 0.41
CDK1 P06493 3/20 0.41
CCNB1 P14635 3/20 0.41
CCNE2 O96020 2/20 0.41
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CCNB2 O95067 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996492 0.90 PDE2A (0.47) PDE2ACCNE1CDK2CDK1CCNB1
SCHEMBL4947310 0.90 PDE2A (0.62) PDE2ACCNE1CDK2CDK1CCNB1
SCHEMBL6991547 0.90 PDE2A (0.49) PDE2ACCNE1CDK2CDK1CCNB1
SCHEMBL6997188 0.90 CCNE2 (0.52) PDE2ACCNE1CDK2CDK1CCNB1
SCHEMBL6998591 0.88 PDE2A (0.45) PDE2AKMT2AKDM4EALDH1A1
SCHEMBL6987730 0.86 GAA (0.43) PDE2AKMT2AKDM4EALDH1A1
SCHEMBL6997472 0.86 KDM4E (0.41) PDE2AKDM4E
SCHEMBL6997368 0.85 CCNE2 (0.51) PDE2ACCNE1CDK2CDK1CCNB1
SCHEMBL6994822 0.82 PDE9A (0.49) PDE2AKMT2A
SCHEMBL6999184 0.81 PDE2A (0.57) PDE2ACCNE1CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973774-B1 1,5-DIHYDRO-PYRAZOLO 3,4-D]-PYRIMIDINONE DERIVATIVES BAYER AG (DE) 2003-01-22 EP disclosed
US-6174884-B1 CARDIOVASCULAR DISORDERS; CEREBROVASCULAR DISEASES; VASCULAR SYSTEM DISORDERS, ESPECIALLY THE PERIPHERAL BLOOD VESSELS; UROGENITAL DISORDERS; HYPOTENSIVE AGENTS; ANTIARRYTHMIA AND -ISCHEMIC AGENTS; PHOSPHODIESTERASE ACTIVITY BAYER AKTIENGESELLSCHAFT (DE) 2001-01-16 US disclosed