SCHEMBL6987730

SCHEMBL6987730

Cc1nn(C(CCCc2ccccc2)C(C)O)c2nc(Cc3ccc(S(=O)(=O)N4CCOCC4)cc3)[nH]c(=O)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 2/20 0.40
PDE2A O00408 3/20 0.39
LMNA P02545 4/20 0.39
HTT P42858 2/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 6/20 0.39
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CASP3 P42574 2/20 0.38
HPGD P15428 1/20 0.37
PDE9A O76083 1/20 0.37
PDE1C Q14123 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998132 0.92 CCNE2 (0.43) GAAATMSMN1; SMN2KDM4ECYP3A4
SCHEMBL1961181 0.87 ALDH1A1 (0.42) GAAATMSMN1; SMN2KDM4ECYP3A4
SCHEMBL6987648 0.86 PDE2A (0.47) KDM4EKMT2APDE2AALDH1A1
SCHEMBL6996492 0.82 PDE2A (0.47) PDE2A
SCHEMBL6998591 0.80 PDE2A (0.45) GAAKDM4EKMT2APDE2ALMNA
SCHEMBL7352650 0.79 ALDH1A1 (0.43) GAAATMSMN1; SMN2KDM4ECYP3A4
SCHEMBL4947310 0.79 PDE2A (0.62) PDE2A
SCHEMBL7885924 0.79 CCNE2 (0.43) GAAATMSMN1; SMN2KDM4ECYP3A4
SCHEMBL6997188 0.77 CCNE2 (0.52) KDM4EKMT2APDE2AALDH1A1
SCHEMBL6991547 0.77 PDE2A (0.49) KDM4EKMT2APDE2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973774-B1 1,5-DIHYDRO-PYRAZOLO 3,4-D]-PYRIMIDINONE DERIVATIVES BAYER AG (DE) 2003-01-22 EP disclosed